崔孙良
教授
个人简介
崔孙良,浙江大学药学院教授、博士生导师 药学院党委委员、院长助理、药物发现与设计研究所所长 中组部“计划”青年拔尖人才 主要从事药物化学的基础研究与新药研发、基于天然产物的新药研发、原料药与医药中间体的新工艺开发等研究工作。以通讯作者发表SCI论文多篇,包括Nature Communications、Angewandte Chemie International Edition、Journal of Medicinal Chemistry等。 教育经历 1999.9—2003.7 浙江大学化学系 本科 2003.9—2008.7 浙江大学化学系 直攻博 2008.9—2010.4 美国科罗拉多州立大学 博士后 2010.5—2012.1 美国南佛罗里达大学 博士后 工作经历 2012.1—2014.12 浙江大学药学院 特聘研究员 2015.1—至今 浙江大学药学院 教授 专利 (1) 崔孙良,张岩,侯廷军,“反式邻羟基二苯乙烯衍生物及其制备方法和应用”,专利号 ZL 201410432114.3 (2) 崔孙良,郑晶,“含有三氟甲基的喹唑啉酮衍生物及其制备方法和应用”,专利号 ZL 201510310121.0 (3) 崔孙良,张岩,郑晶,“一种吲哚或吡咯并嘧啶衍生物的制备方法”,专利号 ZL 201310755538.9 (4) 崔孙良,齐纪凤,“吲唑类化合物及其制备方法和应用”,专利号 ZL 201910299910.7 (5) 崔孙良,曾林伟,“一种N-(吲哚-N-甲酰胺)-α-氨基酰胺衍生物的制备方法”,专利号 ZL 201910520080.6
研究领域
药物化学 有机合成
近期论文
围绕药物化学的基础与应用,开展基于靶标与基于天然产物相结合的药物发现研究,获得了抗癫痫、抗肿瘤等候选化合物。 代表性论文如下 (1) Chengcheng Fan#, Zeyi Zhang#, Zhencheng Lai, Yanzi Yang, Jiaming Li, Lei Liu, Siyu Chen, Xueping Hu, Huajun Zhao*, Sunliang Cui*, Adv. Sci. 2024, 11, 2305432. (2) Shengying Lou, Miaolian Wu*, Sunliang Cui*, Curr. Med. Chem. 2024, 31, 2021-2051. (3) Sunliang Cui*, Linwei Zeng, Nat. Chem. 2023, 15, 597-598. (News & Views) (4) Jiaming Li, Zhencheng Lai, Weiwei Zhang, Linwei Zeng, Sunliang Cui*, Nat. Commun. 2023, 14, 4806-4815. (5) Yongmei Tang#, Fanli Zheng#, Xiaodong Bao, Yanan Zheng, Xueping Hu, Siyue Lou, Huajun Zhao*, Sunliang Cui*, J. Med. Chem. 2023, 66, 11905-11926. (6) Zhencheng Lai, Hao Ni, Xueping Hu, Sunliang Cui*, J. Med. Chem. 2023, 66, 10791-10807. (7) Jiaming Li#, Hongda Sheng#, Yingchao Wang, Zhencheng Lai, Yi Wang*, Sunliang Cui*, J. Med. Chem. 2023, 66, 2946-2963. (8) Linwei Zeng, Fengzhi Zhang*, Sunliang Cui*, Org. Lett. 2023, 25, 443-448. (9) Zhencheng Lai#, Rongkai Wu#, Jiaming Li#, Xing Chen, Linwei Zeng, Xi Wang, Jingjing Guo, Zujin Zhao, Hironao Sajiki, Sunliang Cui*, Nat. Commun. 2022, 13, 435-442. (10) Linwei Zeng#, Jiaming Li#, Sunliang Cui*, Angew. Chem. Int. Ed. 2022, 61, e202205037. (11) Jifeng Qi#, Weihua Wang#, Yongmei Tang#, Shengying Lou, Jiaer Wang, Tao Yuan, Qiaojun He, Bo Yang, Hong Zhu*, Sunliang Cui*, J. Med. Chem. 2022, 65, 3849-3865. (12) Changwei Chen#, Xin Chai#, Xueping Hu#, Shengying Lou, Dan Li*, Tingjun Hou*, Sunliang Cui*, J. Med. Chem. 2022, 65, 13074-13093. (13) Dan Li#, Xiaodong Bao#, Jinping Pang#, Xueping Hu#, Longling Wang#, Jiajia Wang, Zhaoxu Yang, Lei Xu, Siyu Wang, Qinjie Weng*, Sunliang Cui*, Tingjun Hou*, J. Med. Chem. 2022, 65, 15710-15724. (14) Shengying Lou, Sunliang Cui*, Curr. Med. Chem. 2022, 29, 3366-3391. (15) Xianjing Zhou, Linwei Zeng, Yi Wang, Cenglin Xu, Zhong Chen, Sunliang*, Bioorg. Med. Chem. Lett. 2022, 75, 128946-128950. (16) Yanan Li, Chaorong Wang, Tiantian Xu, Peichen Pan, Qing Yu, Xiufang Xiong, Tingjun Hou, Sunliang Cui*, Yi Sun*, Acta Pharm. Sin. B 2021, 11, 3567-3584. (17) Chaorong Wang#, Zhencheng Lai#, Hujun Xie*, Sunliang Cui*, Angew. Chem. Int. Ed. 2021, 60, 5147-5151 (Hot Paper). (18) Zhencheng Lai, Jixiao He, Changxin Zhou, Huajun Zhao, Sunliang Cui*, Curr. Med. Chem. 2021, 28, 2807-2827. (19) Linwei Zeng, Yuxin Lin, Jiaming Li, Hironao Sajiki, Hujun Xie, Sunliang Cui*, Nat. Commun. 2020, 11, 5639-5648. (20) Linwei Zeng, Bo Huang, Yangyong Shen, Sunliang Cui*, Org. Lett. 2018, 20, 3460-3462. (21) Renjie Chen, Linwei Zeng, Bo Huang, Yangyong Shen, Sunliang Cui*, Org. Lett. 2018, 20, 3377-3380. (22) Jifeng Qi, Jing Zheng, Sunliang Cui*, Org. Lett. 2018, 20, 1355-1358. (23) Bo Huang, Linwei Zeng, Yangyong Shen, Sunliang Cui*, Angew. Chem. Int. Ed. 2017, 56, 4565-4568. (24) Yangyong Shen, Bo Huang, Linwei Zeng, Sunliang Cui*, Org. Lett. 2017, 19, 4616-4619. (25) Renjie Chen, Sunliang Cui*, Org. Lett. 2017, 19, 4002-4005. (26) Yangyong Shen, Bo Huang, Jing Zheng, Chen Lin, Yu Liu, Sunliang Cui*, Org. Lett. 2017, 19, 1744-1747. (27) Bo Huang, Linwei Zeng, Yangyong Shen, Sunliang Cui*, Chem. Commun. 2017, 53, 11996-11999. (28) Bo Huang, Yangyong Shen, Zhenjun Mao, Yu Liu, Sunliang Cui*, Org. Lett. 2016, 18, 4888-4891. (29) Yangyong Shen, Jifeng Qi, Zhenjun Mao, Sunliang Cui*, Org. Lett. 2016, 18, 2722-2725. (30) Jing Zheng, Yan Zhang, Dahai Wang, Sunliang Cui*, Org. Lett. 2016, 18, 1768-1771. (31) Jing Zheng, Jifeng Qi, Sunliang Cui*, Org. Lett. 2016, 18, 128-131.