王建武
职称未知
所属大学: 山东大学
所属学院: 化学与化工学院
个人简介
教育 1994-1993: New York University,博士后; 1990-1984: 南开大学,硕士,博士; 1982-1978: 复旦大学,学士; 经历 1999-今: 山东大学化学系,研究员。2001年起,博士生导师; 1999-1998: New York University, 访问教授; 1998-1997: 山东大学化学系, 副教授; 1994-1996: Peptosyn Inc. )研究科学家; 1993-1990: 天津轻工业化学研究所,高工。
研究领域
有机合成:有机合成新反应及新方法。手性合成及功分子合成。天然化合物的全合成及结构修饰; 药物化学:新药物分子设计、合成及构效关系研究,开发新药。
近期论文
Design, synthesis and antibacterial activity of novel actinonin derivatives containing benzimidazole heterocycles, Datong Zhang, Zongheng Wang, Weiren Xu, Fanggang Sun, Lida Tang, Jianwu Wang,, European Journal of Medicinal Chemistry,44 (2009) 2202- 2210 A NOVEL AND EFFICIENT APPROACH TO PYRAZOLO[1,5-a]- PYRIDINE DERIVATIVES VIA ONE-POT TANDEM REACTION, Yan-Qing Ge, Jiong Jia, Yan Li, Ling Yin, and Jianwu Wang* HETEROCYCLES, Vol 78, Issue 1, 2009, pp.197-206 A FACILE APPROACH TO INDOLIZINES VIA TANDEM REACTION, Yan-Qing Ge, Jiong Jia, He Yang, Gui-Long Zhao, Fu-Xu Zhan, and Jianwu Wang*,HETEROCYCLES, Vol. 78, No. 3, 2009, pp. 725 - 736. Polyphosphoric Acid-Mediated, One-Pot, Novel Reactions to Build Polymethoxyarylnaphthalene Lignans,Guilong Zhao a; Fuxu Zhan b; Zhifeng Wang c; Weiren Xu a; Yuli Wang a; Wei Liu a; Lida Tang d;Jianwu Wang b,Synthetic Communications, 1, 40: 351–360, 2010 FACILE SYNTHESIS OF IMIDAZO[1,2-a]PYRIDINES VIA TANDEM REACTION,Jiong Jia,1,2 Yan-Qing Ge,2 Xu-Tang Tao,1*and Jian-Wu Wang2*,HETEROCYCLES, Vol. 81, No. 1, 2010, pp. 185 - 194. Synthesis and antimicrobial activities of novel peptide deformylase inhibitors ,Ling Yin,a Wei-Ren Xu,b Zhi-Guo Wang,c Da-Tong Zhang,a Jiong Jia,a Yan-Qing Ge,aYan Li,a and Jian-Wu Wang a*,ARKIVOC 2010 (ix) 196-205 Synthesis and Preliminary Antibacterial Evaluation of 2-Butyl Succinate-based Hydroxamate Derivatives Containing Isoxazole Rings,Datong Zhang1,2, Jiong Jia1, Lijuan Meng1, Weiren Xu3, Lida Tang3, and Jianwu Wang1,Arch Pharm Res, 2010,0Vol 33, No 6, 831-842. Design,Synthesis and in vivo hypoglycemic activity of tetrazole-bearing N-glycosides as SGLT2 inhibitors, Y L Gao, G L Zhao, W Liu, H Shao, Y L Wang, W R Xu, L D Tang & J W Wang*, Indian Journal of Chemistry, Vol. 49b, November 2010,pp. 1499-1508. The synthesis, characterization and optical properties of novel pyrido[1,2-a]benzimidazole derivatives,Yan Qing Ge a,c,1, Jiong Jia a,b,1, He Yang a, Xu Tang Tao b,*, Jian Wu Wang a,* Dyes and Pigments, 88 (2011), 344-349 Synthesis and optical properties of novel pyrido[1,2-a]benzimidazole-containing 1,3,4-oxadiazole derivatives,He Yang, Yan-Qing Ge, Jiong Jia, Jian-Wu Wang* Journal of Luminescence,131(2011) 749-755 Synthesis, X-ray crystal structure and optical properties of novel 2,5-diaryl-1,3,4-oxadiazole derivatives containing substituted pyrazolo[1,5-a]pyridine units,He Yang, Jinglin Mu, Xia Chen, Lei Feng, Jiong Jia*, Jianwu Wang* Dyes and Pigments,Dyes and PigmentsVolume 91, Issue 3, December 2011, Pages 446-45 Design, synthesis and antibacterial activity of novel N-formylhydroxylamine derivatives as PDF inhibitors,L Yina, J Jiaa, G L Zhaob, W R Xub, L D Tangb & J W Wang*a,Indian Journal of chemistry,2011,50B may, pp695-703 Exquisite Synthesis of a Designed PAR-1 Antagonist, Hua-Ming Miaoa)b), Gui-Long Zhao*b), Lin-Shan Zhangc), Hua Shaob), and Jian-Wu Wang*a) Helvetica Chimica Acta – Vol. 94 (2011) pp 1981-1993 Design and Synthesis of Novel Pyrazole-based Lp-PLA2 Inhibitors Wang, Yia(王毅) Xu, Weirenb(徐为人) Shao, Huab(邵华) Xie, Yafeia(谢亚非) Wang, Jianwu*,a(王建武) Chin. J. Chem. 2011, 29, 2039—2048 The synthesis, characterization and opticalproperties of novel 1,3,4-oxadiazole containing imidazo[1,5-a]pyridinederivatives, Yan Qing Ge a, BenQian Hao a, GuiYun Duan a,, JianWuWang b, Journal of Luminescence 131 (2011) 1070–1076 Design, synthesis and in vivo anti-hyperglycemic activity of gem-dimethyl-bearing C-glucosides as SGLT2 inhibitors. Zhao, Wen Jing; Shi, Yong Heng; Zhao, Gui Long; Wang, Yu Li; Shao, Hua; Li, Da Tang; Wang, Jian Wu. Chinese Chemical Letters (2011), 22(10), 1215-1218. Synthesis and crystal structure ofethyl1-(2-bromoethyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxylate. Wang, Yi; Shao, Hua; Xu, Wei-Ren; Wang, Jian-Wu. Chinese Journal of Structural Chemistry (2012), 31(1), 110-114. Synthesis, X-ray crystal structure and opticalproperties of novel 2-aryl-3-ethoxycarbonyl-4-phenylpyrido[1,2-a]benzimidazoles, Xia Chen,a He Yang,a Yanqing Ge,c Lei Feng,a Jiong Jiaa,b* andJianwu Wanga* Luminescence (2012), 27(5), 382-389 新型咖啡酸五环三萜酯的合成与保肝活性,贾炯, 孙学华, 邵腾飞, 金树根, 高月求, 王建武,有机化学 2012, 32 (04), pp 760-764 From Cyclopropenes to Tetrasubstituted Furans: Tandem Isomerization/Alkenylation Sequence with Cu/Pd Relay Catalysis,Chuanling Song, Lin Ju, Mingchao Wang, Pengcheng Liu, Yuanzhe Zhang, Jianwu Wang,* and Zhenghu Xu*[a], Chem. Eur. J. 2013, 19, 3584 – 3589 A NEW METHOD FOR THE SYNTHESIS OF [1,2,4]TRIAZOLO[1,5-a]-PYRIDINE DERIVATIVES,Wei-Ming Zhao,a Yan-Qing Ge,b* Wei-Ren Xu,c Gui-Long Zhao,c Jiong Jia,a and Jian-Wu Wanga* HETEROCYCLES, Vol. 87, No. 4, 2013, pp. 869-876. SYNTHESIS OF NITROGEN BRIDGEHEAD HETEROCYCLES WITH PHOSPHONATES VIA A NOVEL TANDEM PROCESS,Ya-Fei Xie,a Yan-Qing Ge,a,b Lei Feng,a Hua-Qiang Xu,a Song Meng,a Gui-Long Zhao,c Wei-Ren Xu,c Jiong Jia,a* and Jian-Wu Wanga* HETEROCYCLES, Vol. 87, No. 4, 2013, pp.815-826. FACILE SYNTHESIS OF PYRIDO[1,2-a]BENZIMIDAZOLE DERIVATIVES VIA NOVEL TANDEM REACTION INVOLVING HORNER-EMMONS REACTION,Wen-Jing Zhao,a Ya-Fei Xie,a Yan-Qing Ge,b* Wei-Ren Xu,c Gui-Long Zhao,c and Jian-Wu Wanga*HETEROCYCLES, Vol. 87, No. 5, 2013, pp.1121-1126. Design, synthesis and biological activity of cyclohexane-bearing C-glucoside derivatives as SGLT2 inhibitors, Zhang, Shuo; Wang, Yu-Li; Wei, Qun-Chao; Xu, Wei-Ren; Tang, Li-Da; Zhao, Gui-Long; Wang, Jian-Wu, Chinese Chemical Letters (2013), 24(5), 429-432. Dimerization of cyclopropenes to bifurans using tandem metal relay catalysis† Chuanling Song, Di Sun, Xianglong Peng, Jing Bai, Rongyi Zhang, Shengzhen Hou, Jianwu Wang and Zhenghu Xu* Chem. Commun., 2013, 49, 9167—9169"