项金宝
教授 博导
个人简介
教育背景 2004-2008,吉林大学,化学学院,有机化学,博士(导师:柏旭教授) 2000-2004,吉林大学,化学学院,材料化学,学士 工作经历 2024至今,吉林大学,药学院,院长 2019至今,吉林大学,组合化学与创新药物研究中心,主任 2019至今,吉林大学,药学院,教授/博士生导师 2017-2019,美国斯克利普斯研究所,化学部,访问学者(合作导师:Phil S. Baran院士) 2016-2019,吉林大学,药学院,副教授/博士生导师 2011-2016,吉林大学,药学院,副教授/硕士生导师 2008-2011,吉林大学,药学院,讲师
研究领域
有机电化学合成研究,潜在生物活性骨架的合成方法学研究,天然产物结构修饰与改造,以及相应的创新药物发现和化学生物学研究
近期论文
Xiang, Jinbao#; Shang, Ming#; Kawamata, Yu; Lundberg, Helena; Reisberg, Solomon H; Chen, Miao; Mykhailiuk, Pavel; Beutner, Gregory; Collins, Michael R; Davies, Alyn; Del Bel, Matthew; Gallego, Gary M; Spangler, Jillian E; Starr, Jeremy; Yang, Shouliang; Blackmond, Donna G; Baran, Phil S*; Hindered Dialkyl Ether Synthesis with Electrogenerated Carbocations, Nature, 2019, 573, 398–402.(IF = 50.5,中科院一区论文) Shi, Lingling; Liu, Mian; Zheng, Lianyou; Gao, Qiansong; Wang, Mingchun; Wang, Xin; Xiang, Jinbao*; Electrochemical γ‑Selective Deuteration of Pyridines, Organic Letters, 2024, 26, 4318–4322.(IF = 4.9,中科院一区论文) Xiang, Jinbao#; Wang, Yuji#; Wang, Wanhe; Yu, Jianxin; Zheng, Lianyou; Hong, Yuan; Shi, Lingling; Zhang, Chunling; Chen, Na; Xu, Jia; Gong, Xuelian; Zhang, Zhuoqi; Cui, Hongming; Zhou, Qian; Zhang, Dapeng; Liu, Yanjun; Ke, Ying; Shen, Jingkang; Xia, Guangxin*; Bai, Xu*; Design, Synthesis, and Pharmacological Evaluation of Quinazoline Derivatives as Novel and Potent pan-JAK inhibitors, Bioorganic Chemistry, 2023, 140, 106765.(IF = 4.5,中科院一区论文) Ning, Shulin; Zheng, Lianyou; Gao, Qiansong; Shi, Lingling; Liu, Yueling; Sun, Chengcheng; Zhang, Zhuoqi; Xiang, Jinbao*; New Electrotriggers: p-Methoxycarbonylbenzyl (pMCB) as an Electroremovable Protecting Group for Carboxylic Acids, Phosphoric Acids and Alcohols, Green Chemistry, 2022, 24, 5632–5636.(IF = 9.3,中科院一区论文) Bai, Ya; Shi, Lingling; Zheng, Lianyou; Ning, Shulin; Che, Xin; Zhang, Zhuoqi; Xiang, Jinbao*; Electroselective and Controlled Reduction of Cyclic Imides to Hydroxylactams and Lactams, Organic Letters, 2021, 23, 2298–2302.(IF = 4.9,中科院一区论文)